Vasopressin receptor 1 Antagonists

  • Vasopressin receptor 1
  • Vasopressin receptor 2
Kat.-Nr. Produktname Informationen Selektiv / Pan IC50 / Ki
S2593 Tolvaptan Tolvaptan is an orally effective nonpeptide arginine vasopressin V2 receptor antagonist with IC50 of 3 nM, used to treat hyponatremia. Pan vasopressin receptor 1a, IC50: 580 nM
S2920 Mozavaptan Mozavaptan is a novel competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively. Pan Vasopressin receptor 1, IC50: 1.2 μM
S2116 Conivaptan HCl Conivaptan HCl is a non-peptide inhibitor of antidiuretic hormone (vasopressin receptor antagonist). Pan